Reviews

Progress of small molecules for targeted protein degradation: PROTACs and other technologiesDrug Development Research2023
Novel strategies and promising opportunities for targeted protein degradation: An innovative therapeutic approach to overcome cancer resistancePharmacology and Therapeutics2023
Targeted protein degrader development for cancer: advances, challenges, and opportunitiesTrends in Pharmacological Sciences2023
PROTAC’ing oncoproteins: targeted protein degradation for cancer therapyMolecular Cancer2023
Delivering on the promise of protein degradersNature Reviews Drug Discovery2023
PROTAC targeted protein degraders: the past is prologueNature Reviews Drug Discovery2022
Targeted protein degradation: mechanisms, strategies and applicationSignal Transduction and Targeted Therapy2022
Key Considerations in Targeted Protein Degradation Drug Discovery and DevelopmentFrontiers in Chemistry 2022
Targeted Protein Degradation: Clinical Advances in the Field of OncologyInternational Journal of Molecular Sciences2022
Targeted protein degradation: Emerging concepts and protein state-specific targeting principlesCurrent Opinion in Chemical Biology2022
PROTACs: past, present and futureChemical Society Reviews2022
Protein degradation technology: a strategic paradigm shift in drug discoveryJournal of Hematology and Oncology2021
Small-Molecule Approaches to Targeted Protein DegradationAnnual Reviews of Cancer Biology2021
Molecular Glues for Targeted Protein Degradation: From Serendipity to Rational DiscoveryJournal of Medicinal Chemistry 2021
Recent Developments in PROTAC-Mediated Protein Degradation: From Bench to ClinicChemBioChem2021
Major advances in targeted protein degradation: PROTACs, LYTACs, and MADTACsJournal of Biological Chemistry 2021
The PROTACtable genomeNature Reviews Drug Discovery2021
PROTAC Technology: Opportunities and ChallengesACS Med. Chem. Lett. 2020
PROTACs: An Emerging Therapeutic
Modality in Precision Medicine
Cell Chemical Biology 2020
Targeted protein degradation: expanding the toolboxNature Reviews Drug Discovery2019
Targeted Protein Degradation: from Chemical Biology to Drug DiscoveryCell Chemical Biology2017
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Protein Degraders